3861-3864
| 3 -(4-Ethyl-3-iodophenyl)nortropane-2- carboxylic Acid Methyl Ester as a High-Affinity Selective Ligand for the Serotonin Transporter
Bruce E. Blough,
Philip Abraham,
Andrew C. Mills,
Anita H. Lewin,
John W. Boja,
Ursula Scheffel,
Michael J. Kuhar, and
F. Ivy Carroll
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3865-3868
| Class III Antiarrhythmic Activity in Vivo by Selective Blockade of the Slowly Activating Cardiac Delayed Rectifier Potassium Current IKs by (R)-2-(2,4- Trifluoromethyl)-N-[2-oxo-5-phenyl- 1-(2,2,2-trifluoroethyl)-2,3-dihydro- 1H-benzo[e][1,4]diazepin-3-yl]acetamide
Harold G. Selnick,
Nigel J. Liverton,
John J. Baldwin,
John W. Butcher,
David A. Claremon,
Jason M. Elliott,
Roger M. Freidinger,
Stella A. King,
Brian E. Libby,
Charles J. McIntyre,
David A. Pribush,
David C. Remy,
Garry R. Smith,
Andrew J. Tebben,
Nancy K. Jurkiewicz,
Joseph J. Lynch,
Joseph J. Salata,
Michael C. Sanguinetti,
Peter K. S. Siegl,
Donald E. Slaughter, and
Kamlesh Vyas
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3869-3870
| Potent and Selective Inhibition of Neuronal Nitric Oxide Synthase by N -Propyl-L-arginine
Henry Q. Zhang,
Walter Fast,
Michael A. Marletta,
Pavel Martasek, and
Richard B. Silverman
[Full Article -
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3871-3886
| A New Approach to Docking in the 2-Adrenergic Receptor That Exploits the Domain Structure of G-Protein-Coupled Receptors
Paul R. Gouldson,
Christopher R. Snell, and
Christopher A. Reynolds
[Full Article -
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3887-3896
| Boron-Containing Polyamines as DNA Targeting Agents for Neutron Capture Therapy of Brain Tumors: Synthesis and Biological Evaluation
Jianping Cai,
Albert H. Soloway,
Rolf F. Barth,
Dianne M. Adams,
Joya R. Hariharan,
Iwona M. Wyzlic, and
Krista Radcliffe
[Full Article -
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3897-3904
| Syntheses and Photodynamic Activities of Novel Trisulfonated Zinc Phthalocyanine Derivatives
Svetlana Kudrevich,
Nicole Brasseur,
Carole La Madeleine,
Sandra Gilbert, and
Johan E. van Lier
[Full Article -
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3905-3914
| N-Hydroxyalkyl Derivatives of 3-Phenyltropane and 1-Methylspiro[1H-indoline-3,4'-piperidine]: Vesamicol Analogues with Affinity for Monoamine Transporters
Simon M. N. Efange,
Ashok P. Kamath,
Anil B. Khare,
Mei-Ping Kung,
Robert H. Mach, and
Stanley M. Parsons
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3915-3925
| Tyrosine Kinase Inhibitors. 13. Structure-Activity Relationships for Soluble 7-Substituted 4-[(3-Bromophenyl)amino]pyrido[4,3-d]pyrimidines Designed as Inhibitors of the Tyrosine Kinase Activity of the Epidermal Growth Factor Receptor
Andrew M. Thompson,
Donna K. Murray,
William L. Elliott,
David W. Fry,
James A. Nelson,
H. D. Hollis Showalter,
Bill J. Roberts,
Patrick W. Vincent, and
William A. Denny
[Full Article -
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3926-3936
| New Methodology for Profiling Combinatorial Libraries and Screening Sets: Cleaning Up the Design Process with HARPick
Andrew C. Good and
Richard A. Lewis
[Full Article -
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3937-3946
| Antirhino/Enteroviral Vinylacetylene Benzimidazoles: A Study of Their Activity and Oral Plasma Levels in Mice
Mark J. Tebbe,
Wayne A. Spitzer,
Frantz Victor,
Shawn C. Miller,
Chris C. Lee,
Thomas R. Sattelberg, Sr.,
Emma McKinney, and
Joseph C. Tang
[Full Article -
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3947-3956
| Synthesis and Biological Properties of New Constrained CCK-B Antagonists: Discrimination of Two Affinity States of the CCK-B Receptor on Transfected CHO Cells
Bruno Bellier,
Isabelle McCort-Tranchepain,
Bertrand Ducos,
Sophie Danascimento,
Hervé Meudal,
Florence Noble,
Christiane Garbay, and
Bernard P. Roques
[Full Article -
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3957-3962
| Cyclic Enkephalin Analogues with Exceptional Potency and Selectivity for  -Opioid Receptors
Victor J. Hruby,
Hubert Bartosz-Bechowski,
Peg Davis,
Jirina Slaninova,
Teresa Zalewska,
Dagmar Stropova,
Frank Porreca, and
Henry I. Yamamura
[Full Article -
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3963-3968
| NAcSDKP Analogues Resistant to Angiotensin-Converting Enzyme
Sandrine Gaudron,
Marie-Thérèse Adeline,
Pierre Potier, and
Josiane Thierry
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3969-3973
| Enzymatic Properties of the Unnatural -L-Enantiomers of 2',3'-Dideoxyadenosine and 2',3'-Didehydro-2',3'-dideoxyadenosine
Hélène Pélicano,
Claire Pierra,
Staffan Eriksson,
Gilles Gosselin,
Jean-Louis Imbach, and
Georges Maury
[Full Article -
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3974-3978
| 5-HT1B Receptor Antagonist Properties of Novel Arylpiperazide Derivatives of 1-Naphthylpiperazine
Catherine Jorand-Lebrun,
Petrus J. Pauwels,
Christiane Palmier,
Chantal Moret,
Philippe Chopin,
Michel Perez,
Marc Marien, and
Serge Halazy
[Full Article -
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3979-3985
| Viracept (Nelfinavir Mesylate, AG1343): A Potent, Orally Bioavailable Inhibitor of HIV-1 Protease
Stephen W. Kaldor,
Vincent J. Kalish,
Jay F. Davies, II,
Bhasker V. Shetty,
James E. Fritz,
Krzysztof Appelt,
Jeffrey A. Burgess,
Kristina M. Campanale,
Nickolay Y. Chirgadze,
David K. Clawson,
Bruce A. Dressman,
Steven D. Hatch,
Deborah A. Khalil,
Maha B. Kosa,
Penny P. Lubbehusen,
Mark A. Muesing,
Amy K. Patick,
Siegfried H. Reich,
Kenneth S. Su, and
John H. Tatlock
[Full Article -
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3986-3989
| Effect of Stereochemistry on the Clearance Mechanism of 111In(III)-Labeled D- or L-Benzyldiethylenetriaminepentaacetic Acid
Kim A. Deal and
Michael J. Welch
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3990-3990
| Medicinal and Pharmaceutical Chemistry. By Harkishan Singh and V. K. Kapoor. Vallabh Prakashan Publishers, Delhi. 1996. viii + 671 pp. 19 × 25 cm. ISBN 81-85731-00-4. $70 (Rs 560).
John L. Neumeyer
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3990-3990
| Books of Interest
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